產品屬性：
產品名稱 | Vofopitant dihydrochloride |
規格 | 100mg、250mg、500mg |
貨號 | EY-01Y15821 |
Cas No.: 168266-51-1
別名: N/A
化學名: N/A
分子式: C21H25Cl2F3N6O
分子量: 505.36
溶解度: Soluble in DMSO
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
Vofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist, inhibits [3H]SP binding to the NK1 receptor with pKi values of 9.5 and 10.6 in rat and human membranes respectively, acts as a potential broad-spectrum anti-emetic agent[1].pKi: 9.5 (NK1, rat), 10.6 (NK1, human)[1][1]. Gardner CJ, et al. GR205171: a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity. Regul Pept. 1996 Aug 27;65(1):45-53.
特別提醒公司產品僅供科研使用
